Modifying the lipophilic part of phenylthiazole antibiotics to control their drug-likeness-Reference-Cited by-同舟云学术

Modifying the lipophilic part of phenylthiazole antibiotics to control their drug-likeness

Published:2020-01 Issue: Volume:185 Page:111830
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Hosny Yomna,Abutaleb Nader S.,Omara Mariam^ORCID,Alhashimi Marwa,Elsebaei Mohamed M.^ORCID,Elzahabi Heba S.,Seleem Mohamed N.^ORCID,Mayhoub Abdelrahman S.^ORCID

Funder

Academy of Scientific Research and Technology

JESOUR-D program

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference41 articles.

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4. Drug-like properties and the causes of poor solubility and poor permeability;Lipinski;J. Pharmacol. Toxicol. Methods,2000

5. Generation of a set of simple, interpretable ADMET rules of thumb;Gleeson;J. Med. Chem.,2008

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