Development of cell-permeable peptide-based PROTACs targeting estrogen receptor α
Author:
Funder
National Natural Science Foundation of China
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference36 articles.
1. Protacs: chimeric molecules that target proteins to the Skp1-Cullin-F box complex for ubiquitination and degradation;Sakamoto;Proc. Natl. Acad. Sci. U.S.A.,2001
2. Small-molecule modulation of protein homeostasis;Burslem;Chem. Rev.,2017
3. Targeted degradation of the aryl hydrocarbon receptor by the PROTAC approach: a useful chemical genetic tool;Lee;Chembiochem,2010
4. Small-molecule control of intracellular protein levels through modulation of the ubiquitin proteasome system;Buckley;Angew Chem. Int. Ed. Engl.,2014
5. Protac-induced protein degradation in drug discovery: breaking the rules or just making new ones?;Churcher;J. Med. Chem.,2018
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