Progress in the development of β-lactams as N-Acylethanolamine Acid Amidase (NAAA) inhibitors: Synthesis and SAR study of new, potent N-O-substituted derivatives-Reference-Cited by-同舟云学术

Progress in the development of β-lactams as N-Acylethanolamine Acid Amidase (NAAA) inhibitors: Synthesis and SAR study of new, potent N-O-substituted derivatives

Published:2017-01 Issue: Volume:126 Page:561-575
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Petracca R.,Ponzano S.,Bertozzi S.M.,Sasso O.,Piomelli D.,Bandiera T.,Bertozzi F.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference34 articles.

1. Effects of cannabinoid receptor ligands on LPS-induced pulmonary inflammation in mice;Berdyshev;Life Sci.,1998

2. Acute intracerebroventricular administration of palmitoylethanolamide, an endogenous peroxisome proliferator-activated receptor–alpha agonist, modulates carrageenan-induced paw edema in mice;D'Agostino;J. Pharmacol. Exp. Ther.,2007

3. N-(2-Hydroxyethyl)hexadecanamide is orally active in reducing edema formation and inflammatory hyperalgesia by down-modulating mast cell activation;Mazzari;Eur. J. Pharmacol.,1996

4. Control of pain initiation by endogenous cannabinoids;Calignano;Nature,1998

5. Antinociceptive activity of the endogenous fatty acid amide, palmitylethanolamide;Calignano;Eur. J. Pharmacol.,2001

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