3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties-Reference-Cited by-同舟云学术

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties

Published:2015-04 Issue: Volume:94 Page:45-55
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Meinguet Céline^ORCID,Bruyère Céline,Frédérick Raphaël,Mathieu Véronique,Vancraeynest Christelle,Pochet Lionel,Laloy Julie,Mortier Jérémie,Wolber Gerhard,Kiss Robert,Masereel Bernard,Wouters Johan

Funder

Télévie

FRSM

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference23 articles.

1. Harmine inhibits tumour specific neo-vessel formation by regulating VEGF, MMP, TIMP and pro-inflammatory mediators both in vivo and in vitro;Hamsa;Eur. J. Pharmacol.,2010

2. A natural small molecule harmine inhibits angiogenesis and suppresses tumour growth through activation of p53 in endothelial cells;Dai;PLoS One,2012

3. Harmine induces apoptosis in HepG2 cells via mitochondrial signaling pathway;Cao;Hepatobiliary Pancreat. Dis. Int.,2011

4. The beta-carboline alkaloid harmine inhibits BCRP and can reverse resistance to the anticancer drugs Mitoxantrone and Camptothecin in breast cancer cells;Ma;Phyther. Res.,2010

5. Novel trisubstituted harmine derivatives with original in vitro anticancer activity;Frédérick;J. Med. Chem.,2012

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