Synthesis and biological activity of substituted 2,4-diaminopyrimidines that inhibit Bacillus anthracis-Reference-Cited by-同舟云学术

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Synthesis and biological activity of substituted 2,4-diaminopyrimidines that inhibit Bacillus anthracis

Published:2012-08 Issue: Volume:54 Page:387-396
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Nammalwar Baskar,Bunce Richard A.,Berlin K. Darrell,Bourne Christina R.,Bourne Philip C.,Barrow Esther W.,Barrow William W.

Funder

National Institutes of Allergy and Infectious Diseases

National Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference32 articles.

1. Anthrax as a biological weapon: medical and public health management. Working group on civilian biodefense;Inglesby;JAMA,1999

2. Synthetic and crystallographic studies of a new inhibitor series targeting Bacillus anthracis dihydrofolate reductase;Beierlien;J. Med. Chem.,2008

3. Crystal structure of Bacillus anthracis dihydrofolate reductase with the dihydrophthalazine-based trimethoprim derivative RAB1 provides a structural explanation of potency and selectivity;Bourne;Antimicrob. Agents Chemother.,2009

4. In vitro efficacy of new antifolates against trimethoprim-resistant Bacillus anthracis;Barrow;Antimicrob. Agents Chemother.,2007

5. Antifolate Drugs in Cancer Therapy;Jackson,1999

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