Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids. I. Synthesis and biological evaluation of lipophilic conjugates of tranylcypromine-Reference-Cited by-同舟云学术

Enhancement of drug affinity for cell membranes by conjugation with lipoamino acids. I. Synthesis and biological evaluation of lipophilic conjugates of tranylcypromine

Published:2005-11 Issue:11 Volume:40 Page:1074-1079
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Pignatello Rosario,Puleo Antonina,Guccione Salvatore,Raciti Giuseppina,Acquaviva Rosaria,Campisi Agatina,Ventura Cinzia A.,Puglisi Giovanni

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference15 articles.

1. Drug transfer across the blood-brain barrier and improvement of brain delivery

2. Barriers to remember: brain-targeting chemical delivery systems and Alzheimer's disease

3. Determination of lipophilicity and its use as a predictor of blood–brain barrier penetration of molecular imaging agents

4. A Novel Chemical Approach to Drug Delivery: Lipidic Amino Acid Conjugates

5. Lipoamino Acid Conjugates of Methotrexate with Antitumor Activity

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