Discovery of novel N-aryl-2-trifluoromethyl-quinazoline-4-amine derivatives as the inhibitors of tubulin polymerization in leukemia cells

Author:

Wu Hui,Wang Long-Shan,Li Pei,Yu Jia,Cheng Sha,Yu Gang,Ahmad Mashaal,Meng Xue-Ling,Luo Heng,Xu Bi-Xue

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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4. The discovery of novel indazole derivatives as tubulin colchicine site binding agents that displayed potent antitumor activity both in vitro and in vivo;Cui;Eur. J. Med. Chem.,2020

5. Recurrence of the oxazole motif in tubulin colchicine site inhibitors with anti-tumor activity;Barreca;Eur. J. Med. Chem.,2021

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