Highly-tumor-targeted PAD4 inhibitors with PBA modification inhibit tumors in vivo by specifically inhibiting the PAD4-H3cit-NETs pathway in neutrophils
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference38 articles.
1. Human PAD4 regulates histone arginine methylation levels via demethylimination;Wang;Science,2004
2. PAD enzymes in rheumatoid arthritis: pathogenic effectors and autoimmune targets;Curran;Nat. Rev. Rheumatol.,2020
3. PAD4-dependent citrullination of nuclear translocation of GSK3β promotes colorectal cancer progression via the degradation of nuclear CDKN1A;Luo;Neoplasia,2022
4. NETosis proceeds by cytoskeleton and endomembrane disassembly and PAD4-mediated chromatin decondensation and nuclear envelope rupture;Thiam;Proc. Natl. Acad. Sci. U. S. A.,2020
5. PAD4 deficiency improves bleomycin-induced neutrophil extracellular traps and fibrosis in mouse lung;Suzuki;Am. J. Respir. Cell Mol. Biol.,2020
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