Design and syntheses of a bimolecular STING agonist based on the covalent STING antagonist-Reference-Cited by-同舟云学术

Design and syntheses of a bimolecular STING agonist based on the covalent STING antagonist

Published:2023-03 Issue: Volume:250 Page:115184
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Zang Ruochen^ORCID,Xue Liang,Zhang Meifang,Peng Xiaoyue,Li Xionghao,Du Kaixin,Shi Chuanqin,Liu Yuqian,Lin Yuxi,Han Wenwei,Yu Rilei,Wang Qian,Yang Jinbo,Wang Xin,Jiang Tao

Funder

National Natural Science Foundation of China

Taishan Scholar Foundation of Shandong Province

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference52 articles.

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3. STING-dependent cytosolic DNA sensing mediates innate immune recognition of immunogenic tumors;Woo;Immunity,2014

4. Cutting edge: cGAS is required for lethal autoimmune disease in the trex1-deficient mouse model of aicardi-goutières syndrome;Gray;J. Immunol.,2015

5. Pharmacological modulation of nucleic acid sensors - therapeutic potential and persisting obstacles;Vanpouille-Box;Nat. Rev. Drug Discov.,2019

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