Discovery of novel flavonoid-based CDK9 degraders for prostate cancer treatment via a PROTAC strategy
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
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1. Application and challenges of nitrogen heterocycles in PROTAC linker;European Journal of Medicinal Chemistry;2024-07
2. Discovery of novel co-degradation CK1α and CDK7/9 PROTACs with p53 activation for treating acute myeloid leukemia;Bioorganic Chemistry;2024-06
3. PROTACs in Ovarian Cancer: Current Advancements and Future Perspectives;International Journal of Molecular Sciences;2024-05-07
4. Recent Discovery and Development of Inhibitors that Target CDK9 and Their Therapeutic Indications;Journal of Medicinal Chemistry;2024-04-02
5. Characteristic roadmap of linker governs the rational design of PROTACs;Acta Pharmaceutica Sinica B;2024-04
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