Design, synthesis and biological evaluation of novel indole-benzimidazole hybrids targeting estrogen receptor alpha (ER-α)-Reference-Cited by-同舟云学术

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Design, synthesis and biological evaluation of novel indole-benzimidazole hybrids targeting estrogen receptor alpha (ER-α)

Published:2018-02 Issue: Volume:146 Page:206-219
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Singla Ramit,Gupta Kunj Bihari,Upadhyay Shishir,Dhiman Monisha,Jaitak Vikas

Funder

Department of Science and Technology, New Delhi, India

CSIR

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference36 articles.

1. Mitoxantrone- and folate-TPGS2k conjugate hybrid micellar aggregates to circumvent toxicity and enhance efficiency for breast cancer therapy;Guissi;Mol. Pharm.,2017

2. Discovery of a sulfamate-based steroid sulfatase inhibitor with intrinsic selective estrogen receptor modulator properties;Ouellet;Eur. J. Med. Chem.,2016

3. Synthesis and evaluation of tamoxifen derivatives with a long alkyl side chain as selective estrogen receptor down-regulators;Shoda;Bioorg. Med. Chem.,2015

4. The selective estrogen receptor modulator bazedoxifene inhibits hormone-independent breast cancer cell growth and down-regulates estrogen receptor α and cyclin D1;Lewis-Wambi;Mol. Pharmacol.,2011

5. Estrogen receptors: role in breast cancer;Duffy;Crit. Rev. Clin. Lab. Sci.,2006

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1. Synthesis, crystal structure, Hirshfeld, DFT, molecular docking, dynamics studies, and anti-cancer activity of 1-substituted-2-(4-(diethylamino)-2-hydroxyphenyl)- 1H-benzo[d]imidazole-5-ethyl carboxylates;Journal of Molecular Structure;2024-10

2. Estrogen receptor alpha (ER-α) antagonistic activity of phytoconstituents from Potentilla atrosanguinea and Potentilla fulgens in breast cancer;Fitoterapia;2024-09

3. Five‐ or six‐membered aluminum metallocyclic complexes containing N, N bidentate oxazolinyl‐indolate chelate ring: Synthesis, structural, and catalytic studies;Applied Organometallic Chemistry;2024-08-05

4. Indole Compounds in Oncology: Therapeutic Potential and Mechanistic Insights;Pharmaceuticals;2024-07-10

5. Unlocking therapeutic potential: exploring indole scaffolds and their structural insights as pharmacophores in designing anti-breast cancer agents;Medicinal Chemistry Research;2024-06-12

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