Small-molecule PROTAC degraders of the Bromodomain and Extra Terminal (BET) proteins — A review-Reference-Cited by-同舟云学术

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Small-molecule PROTAC degraders of the Bromodomain and Extra Terminal (BET) proteins — A review

Published:2019-04 Issue: Volume:31 Page:43-51
ISSN:1740-6749
Container-title:Drug Discovery Today: Technologies
language:en
Short-container-title:Drug Discovery Today: Technologies

Author:

Yang Chao-Yie,Qin Chong,Bai Longchuan,Wang Shaomeng

Funder

Breast Cancer Research Foundation

Prostate Cancer Foundation

National Cancer Institute

Publisher

Elsevier BV

Subject

Drug Discovery,Molecular Medicine

Reference87 articles.

1. Protacs: chimeric molecules that target proteins to the Skp1–Cullin–F box complex for ubiquitination and degradation;Sakamoto;Proc Natl Acad Sci U S A,2001

2. Small-molecule PROTACS: new approaches to protein degradation;Toure;Angew Chem Int Ed Engl,2016

3. Targeted intracellular protein degradation induced by a small molecule: en route to chemical proteomics;Schneekloth;Bioorg Med Chem Lett,2008

4. Specific degradation of CRABP-II via cIAP1-mediated ubiquitylation induced by hybrid molecules that crosslink cIAP1 and the target protein;Okuhira;FEBS Lett,2011

5. In vivo knockdown of pathogenic proteins via specific and nongenetic Inhibitor of Apoptosis Protein (IAP)-dependent protein erasers (SNIPERs);Ohoka;J Biol Chem,2017

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