Irreversible inactivation of the beta-adrenoreceptor by a partial agonist. Evidence for selective loss of the agonist high affinity binding sites.
Author:
Publisher
Elsevier BV
Subject
Cell Biology,Molecular Biology,Biochemistry
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1. Covalent Molecular Probes for Class A G Protein-Coupled Receptors: Advances and Applications;ACS Chemical Biology;2015-04-22
2. Carbostyril-based beta-adrenergic agonists: evidence for long lasting or apparent irreversible receptor binding and activation of adenylate cyclase activity in vitro;Naunyn-Schmiedeberg's Archives of Pharmacology;2004
3. Irreversible binding of a carbostyril-based agonist and antagonist to the β-adrenoceptor in DDT1MF-2 cells and rat aorta;British Journal of Pharmacology;1998-05
4. NCS-MPP (4-(2′-METHOXY-PHENYL)-1-[2′-(N-2″-PYRIDYL)-P-Isothiocyanobenzamido]-Ethyl-Piperazine): A high affinity and irreversible 5-HT1A receptor ligand;Life Sciences;1995-12
5. Photoaffinity labeling the beta-adrenergic receptor with an iodoazido derivative of norepinephrine.;Journal of Biological Chemistry;1988-10
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