Quantification of azacitidine incorporation into human DNA/RNA by accelerator mass spectrometry as direct measure of target engagement

Author:

Wang Xiaomin,Vaes Wouter H.J.,van Duijn Esther,Nooijen Irene,Tong Zeen,de Menezes Daniel LopesORCID,Maxwell Stephen E.ORCID

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

Reference26 articles.

1. Evaluation of the bioequivalence and food effect on the bioavailability of CC‑486 (oral azacitidine) tablets in adult patients with cancer;Babiker;Cancer Chemo. Pharm.,2020

2. Vidaza® (Azacitidine) Prescribing Information,2018

3. Vidaza (azacitidine);European Medicines Agency,2016

4. US FDA Approves Oral Azacitidine for Acute Myeloid Leukemia,2020

5. Covalent bond formation, between a DNA-cytosine methyltransferase and DNA containing 5-azacytosine;Santi;Proc. Natl. Acad. Sci.,1984

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