Investigation of atropisomeric transformation of a novel PDE4 inhibitor with tetrahydroisoquinoline-based amide group and its primary study of binding to HSA-Reference-Cited by-同舟云学术

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Investigation of atropisomeric transformation of a novel PDE4 inhibitor with tetrahydroisoquinoline-based amide group and its primary study of binding to HSA

Published:2022-11 Issue: Volume:221 Page:115056
ISSN:0731-7085
Container-title:Journal of Pharmaceutical and Biomedical Analysis
language:en
Short-container-title:Journal of Pharmaceutical and Biomedical Analysis

Author:

Chen Huanhuan,Zhu Tingfei,Sun Ling,Xiang Lili,Han Haiyun,Luo Xiaomin,Chen Dongying

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

Reference31 articles.

1. Recent advances in atropisomerism;Ōki;Top. Stereochem.,1983

2. The challenge of atropisomerism in drug discovery;Clayden;Angew. Chem. Int. Ed.,2009

3. Characterization of the in vitro atropisomeric interconversion rates of an endothelin A antagonist by enantioselective liquid chromatography;Shi;J. Chromatogr. A,2005

4. Discovery and assessment of atropisomers of (±)-lesinurad;Wang;ACS Med. Chem. Lett.,2017

5. Benzoisoquinolinediones as potent and selective inhibitors of BRPF2 and TAF1/TAF1L bromodomains;Bouché;J. Med. Chem.,2017

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