ZrCl4-catalyzed nucleophilic dearomatization of 2-hydroxy-pyrimidines: A concise synthesis of novel 3,4-dihydropyrimidin-2(1H)-ones containing a phosphonic ester group-Reference-Cited by-同舟云学术

ZrCl4-catalyzed nucleophilic dearomatization of 2-hydroxy-pyrimidines: A concise synthesis of novel 3,4-dihydropyrimidin-2(1H)-ones containing a phosphonic ester group

Published:2021-06 Issue: Volume:73 Page:153149
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Li Kang-rui,Meng Fan-jie,Jiang Wen-feng,Shi Lei

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference28 articles.

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2. Dihydropyrimidine calcium channel blockers. 3. 3-Carbamoyl-4-aryl-1,2,3,4-tetrahydro-6-methyl-5-pyrimidinecarboxylic acid esters as orally effective antihypertensive agents

3. Design, Synthesis, Biological Evaluation, and Structure–Activity Relationships of Substituted Phenyl 4-(2-Oxoimidazolidin-1-yl)benzenesulfonates as New Tubulin Inhibitors Mimicking Combretastatin A-4

4. Small Molecule Inhibitor of Mitotic Spindle Bipolarity Identified in a Phenotype-Based Screen

5. A Reexamination of the Mechanism of the Biginelli Dihydropyrimidine Synthesis. Support for an N-Acyliminium Ion Intermediate1

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1. Zirconium Tetrachloride;Encyclopedia of Reagents for Organic Synthesis;2024-07-17

2. Phospha-Mannich reactions of phosphinous acids R₂P–OH and their derivatives;Phosphorus, Sulfur, and Silicon and the Related Elements;2023-07-20

3. Recent progress in the direct phosphorylation of parent heterocycles to construct phosphorylated heterocycles;Chemistry of Heterocyclic Compounds;2023-05

4. Zirconium-Based Catalysts in Organic Synthesis;Topics in Current Chemistry;2022-08-11

5. Synthesis of 3,4-Dihydropyrimidin(thio)one Containing Scaffold: Biginelli-like Reactions;Pharmaceuticals;2022-07-30