Flumazenil-independent positive modulation of γ-aminobutyric acid action by 6-methylflavone at human recombinant α1β2γ2L and α1β2 GABAA receptors
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference29 articles.
1. 6-Methylflavone, a benzodiazepine receptor ligand with antagonistic properties on rat brain and human recombinant GABAA receptors in vitro;Ai;Drug Dev. Res.,1997
2. Pharmacological profile of apigenin, a flavonoid isolated from matricaria chamomilla;Avallone;Biochem. Pharmacol.,2000
3. Multiple roles of protein kinases in the modulation of gamma-aminobutyric acidA receptor function and cell surface expression;Brandon;J. Pharmacol. Ther.,2002
4. GABA-activated ligand gated ion channels: medicinal chemistry and molecular biology;Chebib;J. Med. Chem.,2000
5. Structure–activity relationships and molecular modeling analysis of flavonoids binding to the benzodiazepine site of the rat brain GABAA receptor complex;Dekermendjian;J. Med. Chem.,1999
Cited by 37 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Schisandrin B, a dual positive allosteric modulator of GABAA and glycine receptors, alleviates seizures in multiple mouse models;Acta Pharmacologica Sinica;2023-11-28
2. Anti-neuropathic effect of 7,3′-dihydroxyflavone in paclitaxel induced peripheral neuropathy in mice involving GABAA, KATP channel and adenosine receptors;Neurochemistry International;2022-10
3. Fungal Biotransformation of 2′-Methylflavanone and 2′-Methylflavone as a Method to Obtain Glycosylated Derivatives;International Journal of Molecular Sciences;2021-09-05
4. Anxiolytic–like activity of 5–methoxyflavone in mice with involvement of GABAergic and serotonergic systems - in vivo and in silico evidences;European Neuropsychopharmacology;2020-07
5. Rational approaches for the design of various GABA modulators and their clinical progression;Molecular Diversity;2020-03-13
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3