A novel partial agonist of GPBA reduces blood glucose level in a murine glucose tolerance test

Author:

Enomoto Rina,Kurosawa Aya,Nikaido Yoshiaki,Mashiko Misaki,Saheki Toshihiko,Nakajima Nozomi,Kuroiwa Satoshi,Otobe Michinari,Ohsaki Maki,Tooyama Kazuya,Inoue Yusuke,Kuwabara Nobuo,Kikuchi Osamu,Kitamura Tadahiro,Kojima Itaru,Nakagawa Yuko,Saito Tamio,Osada Hiroyuki,Futahashi Mizuko,Sezutsu Hideki,Takeda Shigeki

Funder

Ministry of Agriculture, Forestry and Fisheries of Japan

Publisher

Elsevier BV

Subject

Pharmacology

Reference23 articles.

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3. Long-term safety and efficacy of fasiglifam (TAK-875), a G-protein-coupled receptor 40 agonist, as monotherapy and combination therapy in Japanese patients with type 2 diabetes: a 52-week open-label phase III study;Kaku;Diabetes,2016

4. A G protein-coupled receptor responsive to bile acids;Kawamata;J. Biol. Chem.,2003

5. GPBA: a GPCR for bile acids and an emerging therapeutic target for disorders of digestion and sensation;Lieu;Br. J. Pharm.,2014

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