The long duration of action of the second generation antihistamine bilastine coincides with its long residence time at the histamine H1 receptor
Author:
Funder
Florida Agricultural Experiment Station
Publisher
Elsevier BV
Subject
Pharmacology
Reference22 articles.
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2. The target residence time of antihistamines determines their antagonism of the G protein-coupled histamine H1 receptor;Bosma;Front. Pharmacol.,2017
3. Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973
4. Comparative inhibition by bilastine and cetirizine of histamine-induced wheal and flare responses in humans;Church;Inflamm. Res.,2011
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