Allosteric effects of R- and S-citalopram on the human 5-HT transporter: Evidence for distinct high- and low-affinity binding sites
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference30 articles.
1. High affinity recognition of serotonin transporter antagonists defined by species-scanning mutagenesis — an aromatic residue in transmembrane domain I dictates species-selective recognition of citalopram and mazindol;Barker;J. Biol. Chem.,1998
2. Synaptic uptake and beyond: the sodium- and chloride-dependent neurotransmitter transporter family SLC6;Chen;Pflugers Arch.,2004
3. The S-enantiomer of R,S-citalopram, increases inhibitor binding to the human serotonin transporter by an allosteric mechanism. Comparison with other serotonin transporter inhibitors;Chen;Eur. Neuropsychopharmacol.,2005
4. Characterization of an allosteric citalopram-binding site at the serotonin transporter;Chen;J. Neurochem.,2005
5. Effects of acute and long-term administration of escitalopram and citalopram on serotonin neurotransmission: an in vivo electrophysiological study in rat brain;EL Mansari;Neuropsychopharmacology,2005
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