Na+ modulation, inverse agonism, and anorectic potency of 4-phenylpiperidine opioid antagonists
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference39 articles.
1. Sodium ions increase the binding of the antagonist peptide ICI 174864 to the delta-opiate receptor;Appelmans;Neuropeptides,1986
2. 3H-Naloxone benzoylhydrazone binding in MOR-1-transfected chinese hamster ovary cells: evidence for G-protein-dependent antagonist binding;Brown;J. Pharmacol. Exp. Ther.,1998
3. Combined blockade of both mu- and kappa-opioid receptors prevents the acute orexigenic action of Agouti-related protein;Brugman;Endocrinology,2002
4. Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 percent inhibition (I50) of an enzymatic reaction;Cheng;Biochem. Pharmacol.,1973
5. Selectivity of ligand binding to opioid receptors in brain membranes from the rat, monkey, and guinea pig;Clark;Eur. J. Pharmacol.,1989
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