A region of N-type Ca2+ channel critical for blockade by the dihydropyridine amlodipine

Author:

Miyashita Yoriko,Furukawa Taiji,Kamegaya Etsuko,Yoshii Mitsunobu,Nukada Toshihide

Publisher

Elsevier BV

Subject

Pharmacology

Reference44 articles.

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2. Long-acting dihydropyridine calcium antagonists. 1. 2-Alkoxymethyl derivatives incorporating basic substituents;Arrowsmith;J. Med. Chem.,1986

3. Calcium channel blocking properties of amlodipine in vascular smooth muscle and cardiac muscle in vitro: evidence for voltage modulation of vascular dihydropyridine receptors;Burges;J. Cardiovasc. Pharmacol.,1987

4. Characterizing the 1, 4-dihydropyridines binding interactions in the L-type Ca2+ channel: model construction and docking calculations;Cosconati;J. Med. Chem.,2007

5. Ataxia, arrhythmia and ion-channel gene defects;Doyle;Trends Genet.,1998

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