DNA gyrase inhibitors: Progress and synthesis of potent compounds as antibacterial agents
Author:
Publisher
Elsevier BV
Subject
Pharmacology,General Medicine
Reference74 articles.
1. Exploiting bacterial DNA gyrase as a drug target: current state and perspectives;Collin;Appl. Microbiol. Biotechnol.,2011
2. DNA topoisomerases: harnessing and constraining energy to govern chromosome topology;Schoeffler;Q. Rev. Biophys.,2008
3. DNA topoisomerase I is involved in both repression and activation of transcription;Merino;Nature,1993
4. Mammalian topoisomerase I has base mismatch nicking activity;Yeh;J. Biol. Chem.,1994
5. Topoisomerase as target for antibacterial and anticancer drug discovery;Kathiravan;J. Enzyme Inhib. Med. Chem.,2013
Cited by 158 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Abietane diterpenoid salvipisone: Structure elucidation, conformational analysis, and antimicrobial activity;Journal of Molecular Structure;2025-02
2. Synthesis and computational studies of new pyridine, pyrazole, pyran, and pyranopyrimidine-based derivatives of potential antimicrobial activity as DNA gyrase and topoisomerase IV inhibitors;Journal of Molecular Structure;2025-01
3. Antimicrobial effects of new tetrahydrofurans;European Journal of Medicinal Chemistry Reports;2024-12
4. Discovery of new molecular hybrid derivatives with coumarin scaffold bearing pyrazole/oxadiazole moieties: Molecular docking, POM analyses, in silico pharmacokinetics and in vitro antimicrobial evaluation with identification of potent antitumor pharmacophore sites;Bioorganic Chemistry;2024-12
5. Recent advances and challenges of revolutionizing drug-resistant tuberculosis treatment;European Journal of Medicinal Chemistry;2024-11
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3