Crystal structure of the HIV-1 integrase core domain in complex with sucrose reveals details of an allosteric inhibitory binding site-Reference-Cited by-同舟云学术

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Crystal structure of the HIV-1 integrase core domain in complex with sucrose reveals details of an allosteric inhibitory binding site

Published:2010-03-12 Issue:8 Volume:584 Page:1455-1462
ISSN:0014-5793
Container-title:FEBS Letters
language:en
Short-container-title:

Author:

Wielens Jerome,Headey Stephen J.,Jeevarajah Dharshini,Rhodes David I.,Deadman John,Chalmers David K.,Scanlon Martin J.,Parker Michael W.

Funder

Australian Research Council Linkage project

Commonwealth of Australia

Publisher

Wiley

Subject

Cell Biology,Genetics,Molecular Biology,Biochemistry,Structural Biology,Biophysics

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1016/j.febslet.2010.03.016/fullpdf

Reference78 articles.

1. Integration;Brown,1997

2. Relationship between the oligomeric status of HIV-1 integrase on DNA and enzymatic activity;Guiot;J. Biol. Chem.,2006

3. Molecular mechanisms of HIV integration and therapeutic intervention;Vandegraaff;Expert Rev. Mol. Med.,2007

4. Discovery of raltegravir, a potent, selective orally bioavailable HIV-integrase inhibitor for the treatment of HIV-AIDS infection;Summa;J. Med. Chem.,2008

5. Treatment of HIV infection with raltegravir;Chirch;Expert Opin. Pharmacother.,2009

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4. Structure of a HIV-1 IN-Allosteric Inhibitor Complex at 2.93 Å Resolution: Routes to Inhibitor Optimization;2022-06-09

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