Asymmetric hydrogenation of tetrahydropyrazines: Synthesis of (S)-piperazine-2-tert-butylcarboxamide, an intermediate in the preparation of the HIV protease inhibitor indinavir-Reference-Cited by-同舟云学术

Asymmetric hydrogenation of tetrahydropyrazines: Synthesis of (S)-piperazine-2-tert-butylcarboxamide, an intermediate in the preparation of the HIV protease inhibitor indinavir

Published:1995-09 Issue:36 Volume:36 Page:6419-6422
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Rossen K.,Weissman Steven A.,Sager J.,Reamer R.A.,Askin D.,Volante R.P.,Reider P.J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference13 articles.

1. Present Status and Future Prospects for HIV Therapies

2. Chapter 14. HIV Protease Inhibitors

3. L-735,524: The Design of a Potent and Orally Bioavailable HIV Protease Inhibitor

4. Diastereoselective syn-epoxidation of 2-alkyl-4-enamides to epoxyamides: Synthesis of the Merck HIV-1 protease inhibitor epoxide intermediate

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