4-Hydroxy-2-methyl-3(2H)-isothiazolone-1,1-dioxide as protecting group of 4-(N-methylaminosulfonyl)methylphenylhydrazine during Fischer indole synthesis-Reference-Cited by-同舟云学术

4-Hydroxy-2-methyl-3(2H)-isothiazolone-1,1-dioxide as protecting group of 4-(N-methylaminosulfonyl)methylphenylhydrazine during Fischer indole synthesis

Published:1995-08 Issue:35 Volume:36 Page:6227-6230
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Remuzon P.,Dussy C.,Jacquet J.P.,Soumeillant M.,Bouzard D.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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1. The development of a highly selective 5-HT1 receptor agonist, sumatriptan, for the treatment of migraine

2. 5-Hydroxtryptamine 1D Receptor Agonism Predicts Antimigraine Efficacy

3. The synthesis of a conformationally restricted analog of the anti-migraine drug sumatriptan

4. Synthesis, biological activity and electrostatic properties of 3-[2-(dimethylamino)ethyl]-5-[(3-amino-1,2,4-thiadiazol-5-yl)methyl]-1H-indole, a novel 5-HT1D receptor agonist.

5. Improved Fischer Indole Reaction for the Preparation of N,N-Dimethyltryptamines: Synthesis of L-695,894, a Potent 5-HT1D Receptor Agonist

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