Highly stereoselective access to novel 2,2,4-substituted tetrahydrofurans by halocyclization: Practical chemoenzymatic synthesis of Sch 51048, a broad-spectrum orally active antifungal agent-Reference-Cited by-同舟云学术

Highly stereoselective access to novel 2,2,4-substituted tetrahydrofurans by halocyclization: Practical chemoenzymatic synthesis of Sch 51048, a broad-spectrum orally active antifungal agent

Published:1995-03 Issue:11 Volume:36 Page:1787-1790
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Saksena Anil K,Girijavallabhan Viyyoor M,Lovey Raymond G,Pike Russell E,Wang Haiyan,Ganguly Ashit K,Morgan Brian,Zaks Alexsey,Puar Mohinder S

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference14 articles.

1. 34th Interscience Conference on Antimicrobial Agents and Chemotherapy (ICAAC),1994

2. Enantioselective synthesis of the optical isomers of broad-spectrum orally active antifungal azoles, Sch 42538 and Sch 45012

3. PPL-catalyzed enzymatic asymmetrization of a 2-substituted prochiral 1,3-diol with remote chiral functionality: Improvements toward synthesis of the eutomers of SCH 45012

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