Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor-Reference-Cited by-同舟云学术

Virtual Ligand Screening of the p300/CBP Histone Acetyltransferase: Identification of a Selective Small Molecule Inhibitor

Published:2010-05 Issue:5 Volume:17 Page:471-482
ISSN:1074-5521
Container-title:Chemistry & Biology
language:en
Short-container-title:Chemistry & Biology

Author:

Bowers Erin M.,Yan Gai,Mukherjee Chandrani,Orry Andrew,Wang Ling,Holbert Marc A.,Crump Nicholas T.,Hazzalin Catherine A.,Liszczak Glen,Yuan Hua,Larocca Cecilia,Saldanha S. Adrian,Abagyan Ruben,Sun Yan,Meyers David J.,Marmorstein Ronen,Mahadevan Louis C.,Alani Rhoda M.,Cole Philip A.

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,General Medicine,Biochemistry

Reference63 articles.

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4. Curcumin, a novel p300/CREB-binding protein-specific inhibitor of acetyltransferase, represses the acetylation of histone/nonhistone proteins and histone acetyltransferase-dependent chromatin transcription;Balasubramanyam;J. Biol. Chem.,2004

5. The CBP co-activator is a histone acetyltransferase;Bannister;Nature,1996

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