Mapping the Binding Site of BMS-708163 on γ-Secretase with Cleavable Photoprobes-Reference-Cited by-同舟云学术

Mapping the Binding Site of BMS-708163 on γ-Secretase with Cleavable Photoprobes

Published:2017-01 Issue:1 Volume:24 Page:3-8
ISSN:2451-9456
Container-title:Cell Chemical Biology
language:en
Short-container-title:Cell Chemical Biology

Author:

Gertsik Natalya,am Ende Christopher W.,Geoghegan Kieran F.,Nguyen Chuong,Mukherjee Paramita,Mente Scot,Seneviratne Uthpala,Johnson Douglas S.,Li Yue-Ming

Funder

NIH

Alzheimer Association

JPB Foundation

MetLife Foundation

MSK Cancer Center Support Grant

Commonwealth Foundation for Cancer Research

Experimental Therapeutics Center of MSKCC

William Randolph Hearst Fund

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

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4. Profiling protein methylation with cofactor analog containing terminal alkyne functionality;Blum;Curr. Protoc. Chem. Biol.,2013

5. Safety and tolerability of the gamma-secretase inhibitor avagacestat in a phase 2 study of mild to moderate Alzheimer disease;Coric;Arch. Neurol.,2012

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