BIBP 3226, a potent and selective neuropeptide Y Y1-receptor antagonist. Structure-activity studies and localization of the human Y1 receptor binding site-Reference-Cited by-同舟云学术

BIBP 3226, a potent and selective neuropeptide Y Y1-receptor antagonist. Structure-activity studies and localization of the human Y1 receptor binding site

Published:1997 Issue: Volume: Page:175-XX
ISSN:
Container-title:Neuropeptide Y and Drug Development
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Author:

Rudolf Klaus,Eberlein Wolfgang,Engel Wolfhard,Beck-Sickinger Annette G.,Wittneben Helmut,Wieland Heike A.,Doods Henri N.

Publisher

Elsevier

Reference28 articles.

1. Characterization of neuropeptide Y (NPY) receptors in human cerebral arteries with selective agonists and the new Y1 antagonist BIBP 3226;Abounader;Br. J. Pharmacol.,1995

2. [d-Trp32] Neuropeptide Y: A competitive antagonist of NPY in rat hypothalamus;Balasubramaniam;J. Med. Chem.,1994

3. Structure-activity relationships of neuropeptide Y analogues with respect to Y1 and Y2 receptors;Beck-Sickinger;Biopolymers,1995

4. Complete L-alanine scan of neuropeptide Y reveals ligands binding to Y1 and Y2 receptors with distinguished conformations;Beck-Sinkinger;Eur. J. Biochem.,1994

5. Pathophysiological role of endothelin revealed by the first orally active endothelin receptor antagonist;Clozel;Nature (Lond.),1993

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