Automation of the radiosynthesis and purification procedures for [18F]Fluspidine preparation, a new radiotracer for clinical investigations in PET imaging of σ1 receptors in brain-Reference-Cited by-同舟云学术

Automation of the radiosynthesis and purification procedures for [18F]Fluspidine preparation, a new radiotracer for clinical investigations in PET imaging of σ1 receptors in brain

Published:2014-02 Issue: Volume:84 Page:1-7
ISSN:0969-8043
Container-title:Applied Radiation and Isotopes
language:en
Short-container-title:Applied Radiation and Isotopes

Author:

Maisonial-Besset Aurélie,Funke Uta,Wenzel Barbara,Fischer Steffen,Holl Katharina,Wünsch Bernhard,Steinbach Jörg,Brust Peter

Publisher

Elsevier BV

Subject

Radiation

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4. Synthesis, pharmacological activity and structure affinity relationships of spirocyclic sigma(1) receptor ligands with a (2-fluoroethyl) residue in 3-position;Große Maestrup;Bioorg. Med. Chem.,2011

5. Evaluation of spirocyclic 3-(3-fluoropropyl)-2-benzofurans as sigma1 receptor ligands for neuroimaging with positron emission tomography;Große Maestrup;J. Med. Chem.,2009

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4. Sigma-1 and dopamine D2/D3 receptor occupancy of pridopidine in healthy volunteers and patients with Huntington disease: a [18F] fluspidine and [18F] fallypride PET study;European Journal of Nuclear Medicine and Molecular Imaging;2020-09-29

5. Short and Atom-Economic Enantioselective Synthesis of the σ1-Receptor Ligands (S)- and (R)-Fluspidine—Important Tools for Positron Emission Tomography Studies;The Journal of Organic Chemistry;2019-09-16