Design, synthesis and computational approach to study novel pyrrole scaffolds as active inhibitors of enoyl ACP reductase (InhA) and Mycobacterium tuberculosis antagonists-Reference-Cited by-同舟云学术

Design, synthesis and computational approach to study novel pyrrole scaffolds as active inhibitors of enoyl ACP reductase (InhA) and Mycobacterium tuberculosis antagonists

Published:2022-11 Issue:11 Volume:99 Page:100674
ISSN:0019-4522
Container-title:Journal of the Indian Chemical Society
language:en
Short-container-title:Journal of the Indian Chemical Society

Author:

Prem Kumar S.R.^ORCID,Shaikh Ibrahim Ahmed,Mahnashi Mater H.,Alshahrani Mohammed Abdulrahman,Dixit Sheshagiri R.,Kulkarni Venkatarao H.,Lherbet Christian,Gadad Andanappa K.,Aminabhavi Tejraj M.,Joshi Shrinivas D.

Publisher

Elsevier BV

Subject

Electrochemistry,Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery

Reference51 articles.

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4. Pharmacophore mapping, molecular docking, chemical synthesis of some novel pyrrolyl benzamide derivatives and evaluation of their inhibitory activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis;Joshi;Bioorg. Chem.,2018

5. Inhibition of Mycobacterium tuberculosis InhA by 3-nitropropanoic acid;Songsiriritthigul;Proteins,2022

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2. Synthesis, molecular docking study and biological evaluation of new pyrrole scaffolds as potential antitubercular agents for dual targeting of enoyl ACP reductase and dihydrofolate reductase;PLOS ONE;2024-05-13

3. Synthesis, Molecular Docking Study, and Biological Evaluation of New 4-(2,5-Dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl)benzohydrazides as Dual Enoyl ACP Reductase and DHFR Enzyme Inhibitors;Antibiotics;2023-04-16

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