Synthesis of an analogue of the substance P C-terminal hexapeptide with modification at the glutaminyl and methioninyl residues and increased activity in NK-2 receptor type: Structure-activity relationships
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference32 articles.
1. Substance P and Neurokinins;Henry,1987
2. Receptors for Substance P and Related Neurokinins
3. A potent and selective agonist for NK-2 tachykinin receptor
4. Pharmacological specificity of synthetic peptides as antagonists at tachykinin receptors
5. Development of NK-2 selective antagonists
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1. Analogues of the C-terminal fragments of neurokinins with modifications at their C-terminal methionyl residue;International Journal of Peptide and Protein Research;2009-01-12
2. Synthesis of potent agonists of Substance P by replacement of Met11 with Glu(OBzl) and N-terminal glutamine with Glp of the C-terminal hexapeptide and heptapeptide of Substance P;International Journal of Peptide and Protein Research;2009-01-12
3. Synthesis and epimerization of phenylalanyl 4-aminocyclophosphamides;Tetrahedron;2007-10
4. Phenylalanyl-aminocyclophosphamides as model prodrugs for proteolytic activation: Synthesis, stability, and stereochemical requirements for enzymatic cleavage;Bioorganic & Medicinal Chemistry Letters;2007-01
5. Synthesis and biological activity of NK1 substance P selective agonists by modifying the methionyl residue;Neuropeptides;1994-07
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