Synthesis of an analogue of the substance P C-terminal hexapeptide with modification at the glutaminyl and methioninyl residues and increased activity in NK-2 receptor type: Structure-activity relationships-Reference-Cited by-同舟云学术

Synthesis of an analogue of the substance P C-terminal hexapeptide with modification at the glutaminyl and methioninyl residues and increased activity in NK-2 receptor type: Structure-activity relationships

Published:1992-12 Issue:9 Volume:27 Page:949-954
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Manolopoulou A,Poulos C,Tsegenidis T

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference32 articles.

1. Substance P and Neurokinins;Henry,1987

2. Receptors for Substance P and Related Neurokinins

3. A potent and selective agonist for NK-2 tachykinin receptor

4. Pharmacological specificity of synthetic peptides as antagonists at tachykinin receptors

5. Development of NK-2 selective antagonists

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