Discovery of a novel series of 6-azauracil-based thyroid hormone receptor ligands: potent, TRβ subtype-selective thyromimetics-Reference-Cited by-同舟云学术

Discovery of a novel series of 6-azauracil-based thyroid hormone receptor ligands: potent, TRβ subtype-selective thyromimetics

Published:2003-02 Issue:3 Volume:13 Page:379-382
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Dow Robert L.,Schneider Steven R.,Paight Ernest S.,Hank Richard F.,Chiang Phoebe,Cornelius Peter,Lee Eunsun,Newsome William P.,Swick Andrew G.,Spitzer Josephine,Hargrove Diane M.,Patterson Terrell A.,Pandit Jayvardhan,Chrunyk Boris A.,LeMotte Peter K.,Danley Dennis E.,Rosner Michele H.,Ammirati Mark J.,Simons Samuel P.,Schulte Gayle K.,Tate Bonnie F.,DaSilva-Jardine Paul

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference10 articles.

1. METABOLIC ASPECTS OF THE CALORIGENIC EFFECT OF THYROID HORMONE IN MAMMALS

2. Species Differences in Cardiac Thyroid Hormone Receptor Isoforms Protein Abundance.

3. Thyroxine analogs. XIX. 3,5-Dimethyl-3'-isopropyl-DL-thyronine

4. A high-affinity subtype-selective agonist ligand for the thyroid hormone receptor

5. A Subtype-Selective Thyromimetic Designed to Bind a Mutant Thyroid Hormone Receptor Implicated in Resistance to Thyroid Hormone

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