The rational development of small molecule tachykinin NK3 receptor selective antagonists - the utilisation of a dipeptide chemical library in drug design-Reference-Cited by-同舟云学术

The rational development of small molecule tachykinin NK3 receptor selective antagonists - the utilisation of a dipeptide chemical library in drug design

Published:1994-07 Issue:14 Volume:4 Page:1679-1684
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Boden P.,Eden J.M.,Hodgson J.,Horwell D.C.,Howson W.,Hughes J.,McKnight A.T.,Meecham K.,Pritchard M.C.,Raphy J.,Ratcliffe G.S.,Suman-Chauhan N.,Woodruff G.N.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. A new type of synthetic peptide library for identifying ligand-binding activity

2. A general and expedient method for the solid-phase synthesis of 1,4-benzodiazepine derivatives

3. The design of a dipeptide library for screening at peptide receptor sites

4. Rationally designed "dipeptoid" analogs of CCK. .alpha.-Methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolytic properties

5. Design of Specific Inhibitors of Angiotensin-Converting Enzyme: New Class of Orally Active Antihypertensive Agents

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