The design, synthesis and physical chemical properties of novel human vasopressin V 2 -receptor antagonists optimized for parenteral delivery-Reference-Cited by-同舟云学术

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The design, synthesis and physical chemical properties of novel human vasopressin V 2 -receptor antagonists optimized for parenteral delivery

Published:2000-04 Issue:8 Volume:10 Page:783-786
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ashwell M.A,Bagli J.F,Caggiano T.J,Chan P.S,Molinari A.J,Palka C,Park C.H,Rogers J.F,Sherman M,Trybulski E.J,Williams D.K

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference12 articles.

1. 5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]- [1,4]benzodiazepin-10(11H)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985): An Orally Active Arginine Vasopressin Antagonist with Selectivity for V2 Receptors

2. For general principles see Yalkowsky, S. H. Solubility and Solubilization in Aqueous Media; Oxford University Press: New York, 1999.

3. 4,10-dihydro-5H-thieno[3,2-c][1]benzazepine derivatives and 9,10-dihydro-4H-thieno[2,3-c][1]benzazepine derivatives as orally active arginine vasopressin receptor antagonists

Cited by 14 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Discovery of Nonpeptide Vasopressin V2 Receptor Antagonists;Analogue-Based Drug Discovery III;2012-12-18

2. Assessment of Exposure of Metabolites in Preclinical Species and Humans at Steady State from the Single-Dose Radiolabeled Absorption, Distribution, Metabolism, and Excretion Studies: A Case Study;Drug Metabolism and Disposition;2012-04-03

3. ChemInform Abstract: The Design, Synthesis, and Physical Chemical Properties of Novel Human Vasopressin V2-Receptor Antagonists Optimized for Parenteral Delivery.;ChemInform;2010-06-07

4. Synthesis and evaluation of azabicyclo[3.2.1]octane derivatives as potent mixed vasopressin antagonists;Bioorganic & Medicinal Chemistry Letters;2010-06

5. Tricyclic Structures in Medicinal Chemistry: An Overview of their Recent Uses in Non-CNS Pathologies;Mini-Reviews in Medicinal Chemistry;2008-12-01

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