Use of CoMFA in validating the conformation used in designing 4-(1H-benzimidazole-2-carbonyl)piperidines with H1/NK1 receptor antagonist activity-Reference-Cited by-同舟云学术

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Use of CoMFA in validating the conformation used in designing 4-(1H-benzimidazole-2-carbonyl)piperidines with H1/NK1 receptor antagonist activity

Published:1997-11 Issue:22 Volume:7 Page:2825-2830
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Vaz Roy J,Maynard George D,Kudlacz Elizabeth M,Bratton Larry D,Kane John M,Shatzer Scott A,Knippenberg Robert W

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference13 articles.

1. Identification and chemical synthesis of MDL 105,212, a non-peptide tachykinin antagonist with high affinity for NK1 and NK2 receptors

2. A highly convergent synthesis of benzimidazolylpiperidines

3. A potent and selective non-peptide antagonist of the neurokinin a (NK2) receptor

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2. Molecular Docking and Receptor-Based 3D-QSAR Studies on Aromatic Thiazine Derivatives as Selective Aldose Reductase Inhibitors;Acta Physico-Chimica Sinica;2015

3. Chapter 10. The Challenges of Multi-Target Lead Optimization;Drug Discovery;2012

4. Molecular Docking and 3D-QSAR on Maleimide Derivatives as Glycogen Synthase Kinase-3β Inhibitors;Acta Physico-Chimica Sinica;2009

5. Synthesis of substituted 3-arylpiperidines and 3-arylpyrrolidines by radical 1,4 and 1,2-aryl migrations;Tetrahedron;2007-07

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