Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation-Reference-Cited by-同舟云学术

Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation

Published:2015-11 Issue:21 Volume:23 Page:7053-7060
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Ettari Roberta,Pinto Andrea,Previti Santo,Tamborini Lucia,Angelo Ilenia C.,La Pietra Valeria,Marinelli Luciana,Novellino Ettore,Schirmeister Tanja,Zappalà Maria,Grasso Silvana,De Micheli Carlo,Conti Paola

Funder

MIUR

Ministero degli Affari Esteri

DFG

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference42 articles.

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2. The trypanosomiases

3. http://www.who.int/mediacentre/factsheets/fs259/en/.

4. Inhibition of Rhodesain as a Novel Therapeutic Modality for Human African Trypanosomiasis

5. Vinyl Sulfones as Antiparasitic Agents and a Structural Basis for Drug Design

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