Synthesis and characterization of [125I]2-iodo N-[(S)-{(S)-1-methylpiperidin-2-yl}(phenyl)methyl]3-trifluoromethyl-benzamide as novel imaging probe for glycine transporter 1-Reference-Cited by-同舟云学术

Synthesis and characterization of [125I]2-iodo N-[(S)-{(S)-1-methylpiperidin-2-yl}(phenyl)methyl]3-trifluoromethyl-benzamide as novel imaging probe for glycine transporter 1

Published:2011-11 Issue:21 Volume:19 Page:6245-6253
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Fuchigami Takeshi,Haratake Mamoru,Magata Yasuhiro,Haradahira Terushi,Nakayama Morio

Funder

Ichiro Kanehara Foundation

Japan Society for the Promotion of Science (JSPS)

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. Glycine receptors: recent insights into their structural organization and functional diversity

2. Glycine transporters and synaptic function

3. Neurotransmitter transporters expressed in glial cells as regulators of synapse function

4. Glutamate as a therapeutic target in psychiatric disorders

5. Glycine Transporter Inhibitors as Therapeutic Agents for Schizophrenia

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