Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO)-Reference-Cited by-同舟云学术

Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO)

Published:2020-06 Issue:12 Volume:28 Page:115548
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Patnaik Anup,Axford Laura,Deng Lin,Cohick Evan,Ren Xianglin,Loi Sally,Kecman Sam,Hollis-Symynkywicz Micah,Harrison Tyler J.,Papillon Julien P.N.,Dales Natalie,Hamann Lawrence G.,Lee Lac,Regard Jean B.,Marcinkeviciene Jovita,Marro Martin L.,Patterson Andrew W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference42 articles.

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3. Myeloperoxidase: An oxidative pathway for generating dysfunctional high-density lipoprotein;Shao;Chem Res Toxicol,2010

4. Class B scavenger receptors CD36 and SR-BI are receptors for hypochlorite-modified low density lipoprotein;Marsche;J Biol Chem,2003

5. Myeloperoxidase, a leukocyte-derived vascular NO oxidase;Eiserich;Science,2002

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