One-pot synthesis of thioxo-tetrahydropyrimidine derivatives as potent β-glucuronidase inhibitor, biological evaluation, molecular docking and molecular dynamics studies-Reference-Cited by-同舟云学术

One-pot synthesis of thioxo-tetrahydropyrimidine derivatives as potent β-glucuronidase inhibitor, biological evaluation, molecular docking and molecular dynamics studies

Published:2020-04 Issue:7 Volume:28 Page:115359
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Iraji Aida,Nouri Ali,Edraki Najmeh,Pirhadi Somayeh,Khoshneviszadeh Mahsima,Khoshneviszadeh Mehdi

Funder

Shiraz University of Medical Sciences

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

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3. Synthesis and β-glucuronidase inhibitory activity of 2-arylquinazolin-4 (3H)-ones;Khan;Bioorg Med Chem,2014

4. Biology-oriented drug synthesis (BIODS): In vitro β-glucuronidase inhibitory and in silico studies on 2-(2-methyl-5-nitro-1H-imidazol-1-yl) ethyl aryl carboxylate derivatives;Salar;Eur J Med Chem,2017

5. Dihydropyrimidones: As novel class of β-glucuronidase inhibitors;Ali;Bioorg Med Chem,2016

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