Synthesis, structure–activity relationships, and anticonvulsant activities of 2-amino-4H-pyrido[3,2-e][1,3]thiazin-4-one derivatives as orally active AMPA receptor antagonists-Reference-Cited by-同舟云学术

Synthesis, structure–activity relationships, and anticonvulsant activities of 2-amino-4H-pyrido[3,2-e][1,3]thiazin-4-one derivatives as orally active AMPA receptor antagonists

Published:2015-04 Issue:8 Volume:23 Page:1788-1799
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Inami Hiroshi,Shishikura Jun-ichi,Yasunaga Tomoyuki,Ohno Kazushige,Yamashita Hiroshi,Kato Kota,Sakamoto Shuichi

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference42 articles.

1. The Role of Excitotoxicity in Neurodegenerative Disease

2. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

3. Glutamatergic Neurotransmission As Molecular Target of New Anticonvulsants

4. Competitive AMPA receptor antagonists

5. α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Antagonists: From Bench to Bedside

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