Design, synthesis and biological evaluation of bis(hydroxyphenyl) azoles as potent and selective non-steroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) for the treatment of estrogen-dependent diseases-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of bis(hydroxyphenyl) azoles as potent and selective non-steroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) for the treatment of estrogen-dependent diseases

Published:2008-06 Issue:12 Volume:16 Page:6423-6435
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Bey Emmanuel,Marchais-Oberwinkler Sandrine,Kruchten Patricia,Frotscher Martin,Werth Ruth,Oster Alexander,Algül Oztekin,Neugebauer Alexander,Hartmann Rolf W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference79 articles.

1. Oestrogen exposure and breast cancer risk

2. Endometriosis: Role of Ovarian Steroids in Initiation, Maintenance, and Suppression

3. Hormonal therapy for postmenopausal breast cancer: the science of sequencing

4. Advances in Hormonal Therapy for Breast Cancer

5. Overview and new strategies in metastatic breast cancer (MBC) for treatment of tamoxifen-resistant patients

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