Structure activity relationship of selective GABA uptake inhibitors-Reference-Cited by-同舟云学术

Structure activity relationship of selective GABA uptake inhibitors

Published:2015-05 Issue:10 Volume:23 Page:2480-2488
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Vogensen Stine B.,Jørgensen Lars,Madsen Karsten K.,Jurik Andreas,Borkar Nrupa,Rosatelli Emiliano,Nielsen Birgitte,Ecker Gerhard F.,Schousboe Arne,Clausen Rasmus P.

Funder

Lundbeck Foundation

Austrian Science Fund

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

1. Neurotransmitters, Seizures, and Epilepsy III;Nistico,1986

2. GABA-Ergic Drugs: Exit Stage Left, Enter Stage Right

3. Selective GABA Transporter Inhibitors Tiagabine and EF1502 Exhibit Mechanistic Differences in Their Ability to Modulate the Ataxia and Anticonvulsant Action of the Extrasynaptic GABAAReceptor Agonist Gaboxadol

4. Synaptic and extrasynaptic GABA transporters as targets for anti-epileptic drugs

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