Kinetic and docking studies of phenol-based inhibitors of carbonic anhydrase isoforms I, II, IX and XII evidence a new binding mode within the enzyme active site-Reference-Cited by-同舟云学术

Kinetic and docking studies of phenol-based inhibitors of carbonic anhydrase isoforms I, II, IX and XII evidence a new binding mode within the enzyme active site

Published:2011-02 Issue:4 Volume:19 Page:1381-1389
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Durdagi Serdar,Şentürk Murat,Ekinci Deniz,Balaydın Halis Türker,Göksu Süleyman,Küfrevioğlu Ö. İrfan,Innocenti Alessio,Scozzafava Andrea,Supuran Claudiu T.

Funder

7th framework EU programme (Metoxia)

Scientific and Technological Research Council of Turkey

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference51 articles.

1. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

2. Carbonic anhydrase inhibitors

3. Carbonic anhydrases as targets for medicinal chemistry

4. Solvent-Mediated Proton Transfer in Catalysis by Carbonic Anhydrase

5. Bidentate Zinc Chelators for α-Carbonic Anhydrases that Produce a Trigonal Bipyramidal Coordination Geometry

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