Synthesis, docking simulation, biological evaluations and 3D-QSAR study of 5-Aryl-6-(4-methylsulfonyl)-3-(metylthio)-1,2,4-triazine as selective cyclooxygenase-2 inhibitors-Reference-Cited by-同舟云学术

Synthesis, docking simulation, biological evaluations and 3D-QSAR study of 5-Aryl-6-(4-methylsulfonyl)-3-(metylthio)-1,2,4-triazine as selective cyclooxygenase-2 inhibitors

Published:2014-01 Issue:2 Volume:22 Page:865-873
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Irannejad Hamid,Kebriaieezadeh Abbas,Zarghi Afshin,Montazer-Sadegh Farhad,Shafiee Abbas,Assadieskandar Amir,Amini Mohsen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Nonsteroid drug selectivities for cyclo-oxygenase-1 rather than cyclo-oxygenase-2 are associated with human gastrointestinal toxicity: A full in vitro analysis

2. Cyclooxygenase Isozymes: The Biology of Prostaglandin Synthesis and Inhibition

3. Expression of COX-1 and COX-2 in a Clinical Model of Acute Inflammation

4. New insights into eicosanoid biosynthetic pathways: implications for arthritis

Cited by 55 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A structure-based approach to explore novel COX-2 inhibitors using pharmacophore modelling, 3D-QSAR analysis, virtual screening and dynamics simulation study;Journal of Molecular Structure;2024-01

2. Diphenyl-substituted triazine derivatives: synthesis, α-glucosidase inhibitory activity, kinetics and in silico studies;Future Medicinal Chemistry;2023-09

3. Synthesis and Biological Activities of Some 3,5-Disubstituted-6-Oxo-1,2,4-Triazine-2-Thiocarboxamide Derivatives as Anti-Breast Cancer (MCF) and α-Glucosidase Inhibitors;Russian Journal of Bioorganic Chemistry;2023-07-10

4. Synthesis, Reactivity, and Anticancer Activity Evaluation of 4‐Amino‐3‐Mercapto‐6‐Methyl‐1,2,4‐Triazin‐5(4H)‐One Derivatives;ChemistrySelect;2023-05-22

5. Design and Development of COX-II Inhibitors: Current Scenario and Future Perspective;ACS Omega;2023-05-09