Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2-Reference-Cited by-同舟云学术

Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2

Published:2018-07 Issue:11 Volume:26 Page:2965-2972
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Moustakim Moses^ORCID,Riedel Kerstin^ORCID,Schuller Marion,Gehring Andrè P.,Monteiro Octovia P.,Martin Sarah P.,Fedorov Oleg,Heer Jag,Dixon Darren J.,Elkins Jonathan M.,Knapp Stefan,Bracher Franz^ORCID,Brennan Paul E.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference42 articles.

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2. Macrodomains: Structure, Function, Evolution, and Catalytic Activities;Rack;Annu Rev Biochem,2016

3. Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors;Wahlberg;Nat Biotech,2012

4. Substrate-Assisted Catalysis by PARP10 Limits Its Activity to Mono-ADP-Ribosylation;Kleine;Mol Cell,2008

5. The PARP superfamily;Ame;BioEssays,2004

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