Structure-based drug design of novel and highly potent pyruvate dehydrogenase kinase inhibitors-Reference-Cited by-同舟云学术

Structure-based drug design of novel and highly potent pyruvate dehydrogenase kinase inhibitors

Published:2021-12 Issue: Volume:52 Page:116514
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Bessho Yuki,Akaki Tatsuo,Hara Yoshinori,Yamakawa Maki,Obika Shingo,Mori Genki,Ubukata Minoru,Yasue Katsutaka,Nakane Yoshitomi,Terasako Yasuo,Orita Takuya,Doi Satoki,Iwanaga Tomoko,Fujishima Ayumi,Adachi Tsuyoshi,Ueno Hiroshi,Motomura Takahisa

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

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4. Microenvironmental control of glucose metabolism in tumors by regulation of pyruvate dehydrogenase;Golias;Int J Cancer.,2019

5. Cloning and characterization of PDK4 on 7q21.3 encoding a fourth pyruvate dehydrogenase kinase isoenzyme in human;Rowles;J Biol Chem.,1996

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