Identification of novel thiazolo[5,4-d]pyrimidine derivatives as human A1 and A2A adenosine receptor antagonists/inverse agonists
Author:
Funder
University of Florence
University of Ferrara
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
Reference38 articles.
1. International union of basic and clinical pharmacology. LXXXI. Nomenclature and classification of adenosine receptor. An update;Fredholm;Pharmacol Rev,2011
2. Adenosine as a multi-signalling guardian angel in human diseases: when, where and how does it exert its protective effects?;Borea;Trends Pharmacol Sci,2016
3. Adenosine receptors in health and disease;Gessi;Adv Pharmacol,2011
4. Biochemical and pharmacological role of A1 adenosine receptors and their modulation as novel therapeutic strategy;Varani;Adv Exp Med Biol-Protein Rev,2017
5. Adenosine A1 receptor antagonists in clinical research and development;Hocher;Kidney Int,2010
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