Design, synthesis, molecular docking and biological evaluation of thiophen-2-iminothiazolidine derivatives for use against Trypanosoma cruzi-Reference-Cited by-同舟云学术

Design, synthesis, molecular docking and biological evaluation of thiophen-2-iminothiazolidine derivatives for use against Trypanosoma cruzi

Published:2016-09 Issue:18 Volume:24 Page:4228-4240
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Silva-Júnior E.F.,Silva E.P.S.,França P.H.B.,Silva J.P.N.,Barreto E.O.,Silva E.B.,Ferreira R.S.,Gatto C.C.,Moreira D.R.M.,Siqueira-Neto J.L.,Mendonça-Júnior F.J.B.,Lima M.C.A.,Bortoluzzi J.H.,Scotti M.T.,Scotti L.,Meneghetti M.R.,Aquino T.M.,Araújo-Júnior J.X.

Funder

Conselho Nacional de Desenvolvimento Científico e Tecnológico

Coordernação de Aperfeiçoamento de Pessoal de Nível Superior

Fundação de Amparo à Pesquisa do Estado de Alagoas

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

1. Conformational restriction of aryl thiosemicarbazones produces potent and selective anti-Trypanosoma cruzi compounds which induce apoptotic parasite death

2. Design, synthesis and biological evaluation of hybrid bioisoster derivatives of N-acylhydrazone and furoxan groups with potential and selective anti-Trypanosoma cruzi activity

3. Novel nitro(triazole/imidazole)-based heteroarylamides/sulfonamides as potential antitrypanosomal agents

4. Thiosemicarbazones derived from 1-indanones as new anti-Trypanosoma cruzi agents

5. 2-Pyridyl thiazoles as novel anti-Trypanosoma cruzi agents: Structural design, synthesis and pharmacological evaluation

Cited by 44 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. SYNTHESIS AND INVESTIGATION OF α-RHODANOCARBONYL COMPOUNDS;Современные технологии. Технические и естественные науки: сборник статей международной научной конференции (Архангельск, Июнь 2024);2024-08-15

2. A consensus reverse docking approach for identification of a competitive inhibitor of acetyltransferase enhanced intracellular survival protein from Mycobacterium tuberculosis;Bioorganic & Medicinal Chemistry;2024-06

3. Trypanocidal potential of synthetic p-aminochalcones: In silico and in vitro evaluation;Bioorganic Chemistry;2023-12

4. Discovery of Novel Inhibitors of Cruzain Cysteine Protease of Trypanosoma cruz;Current Medicinal Chemistry;2023-10-06

5. One‐Pot Access to Tetrasubstituted 2‐Aminothiophenes via Regio‐ and Chemoselective Domino Reactions of Dithioesters with Fumaronitrile at Room Temperature;Advanced Synthesis & Catalysis;2023-08